Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects
Bioorganic Chemistry, cilt.83, ss.170-179, 2019 (SCI-Expanded, Scopus)
- Yayın Türü: Makale / Tam Makale
- Cilt numarası: 83
- Basım Tarihi: 2019
- Doi Numarası: 10.1016/j.bioorg.2018.10.042
- Dergi Adı: Bioorganic Chemistry
- Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
- Sayfa Sayıları: ss.170-179
- Anahtar Kelimeler: 1,2,4-Triazoles, Carbonic anhydrase, Inhibition, Molecular docking, Uncompetitive, ADME properties, ISOZYME-II, BIOLOGICAL EVALUATION, CRYSTAL-STRUCTURE, DRUG DISCOVERY, X-RAY, SULFONAMIDES, TARGET, IX, TRANSMEMBRANE, DOCKING
- Karadeniz Teknik Üniversitesi Adresli: Evet